AZ4800 [Ligand Id: 7805] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL2151176
  • presenilin 1 in Human [GtoPdb: 2402] [UniProtKB: P49768]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
presenilin 1 in Human [GtoPdb: 2402] [UniProtKB: P49768]
GtoPdb - - 7.59 pIC50 26 nM IC50 J Biol Chem (2012) 287: 11810-9 [PMID:22334705]

ChEMBL data shown on this page come from version 31:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, CibriƔn-Uhalte E, Davies M, Dedman N, Karlsson A, MagariƱos MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]