PFI-3 [Ligand Id: 7915] activity data from GtoPdb

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  • polybromo 1 in Human [GtoPdb: 2738] [UniProtKB: Q86U86]
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  • SWI/SNF related, matrix associated, actin dependent regulator of chromatin, subfamily a, member 4 in Human [GtoPdb: 2740] [UniProtKB: P51532]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
polybromo 1 in Human [GtoPdb: 2738] [UniProtKB: Q86U86]
GtoPdb - - 7.32 pKd 48 nM Kd PFI-3 A Selective chemical probe for SMARCA bromodomains.. thesgc.org
SWI/SNF related, matrix associated, actin dependent regulator of chromatin, subfamily a, member 4 in Human [GtoPdb: 2740] [UniProtKB: P51532]
GtoPdb - - 7.05 pKd 89 nM Kd PFI-3 A Selective chemical probe for SMARCA bromodomains.. thesgc.org

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.