CRT 0066101 [Ligand Id: 8048] activity data from GtoPdb

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  • protein kinase D1 in Human [GtoPdb: 1489] [UniProtKB: Q15139]
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  • protein kinase D2 in Human [GtoPdb: 2173] [UniProtKB: Q9BZL6]
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  • protein kinase D3 in Human [GtoPdb: 2174] [UniProtKB: O94806]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
protein kinase D1 in Human [GtoPdb: 1489] [UniProtKB: Q15139]
GtoPdb - - 9 pIC50 1 nM IC50 Mol Cancer Ther (2010) 9: 1136-46 [PMID:20442301]
protein kinase D2 in Human [GtoPdb: 2173] [UniProtKB: Q9BZL6]
GtoPdb - - 8.6 pIC50 2.5 nM IC50 Mol Cancer Ther (2010) 9: 1136-46 [PMID:20442301]
protein kinase D3 in Human [GtoPdb: 2174] [UniProtKB: O94806]
GtoPdb - - 8.7 pIC50 2 nM IC50 Mol Cancer Ther (2010) 9: 1136-46 [PMID:20442301]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.