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ChEMBL ligand: CHEMBL1084942 |
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DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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BB3 receptor/Bombesin receptor subtype-3 in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL4080] [GtoPdb: 40] [UniProtKB: P32247] | ||||||||
ChEMBL | Agonistic activity at human BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assay | F | 6.88 | pEC50 | 133 | nM | EC50 | Bioorg. Med. Chem. Lett. (2010) 20: 1913-1917 [PMID:20167483] |
BB3 receptor/Bombesin receptor subtype-3 in Mouse (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL1075140] [GtoPdb: 40] [UniProtKB: O54798] | ||||||||
GtoPdb | - | - | 8.59 | pKd | 2.6 | nM | Kd | Cell Metab (2010) 11: 101-12 [PMID:20096642] |
ChEMBL | Agonistic activity at mouse BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assay | F | 8.1 | pEC50 | 7.9 | nM | EC50 | Bioorg. Med. Chem. Lett. (2010) 20: 1913-1917 [PMID:20167483] |
ChEMBL data shown on this page come from version 31:
Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, CibriƔn-Uhalte E, Davies M, Dedman N, Karlsson A, MagariƱos MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]