ChEMBL ligand: CHEMBL420783 (L-740093)
CCK1 receptor/Cholecystokinin A receptor in Rat [ChEMBL: CHEMBL2871] [GtoPdb: 76] [UniProtKB: P30551] There should be some charts here, you may need to enable JavaScript!
CCK2 receptor/Cholecystokinin B receptor in Human [ChEMBL: CHEMBL298] [GtoPdb: 77] [UniProtKB: P32239] There should be some charts here, you may need to enable JavaScript!

DB	Assay description	Assay Type	Standard value	Standard parameter	Original value	Original units	Original parameter	Reference
CCK1 receptor/Cholecystokinin A receptor in Rat (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL2871] [GtoPdb: 76] [UniProtKB: P30551]
GtoPdb	-	-	5.8	pKi	-	-	-	Mol Pharmacol (1994) 46: 943-8 [PMID:7969084]
ChEMBL	Displacement of [125I]-BH CCK-8S from Cholecystokinin type A receptor in rat pancreas	B	5.79	pIC50	1604	nM	IC50	Bioorg. Med. Chem. Lett. (1995) 5: 3023-3026
ChEMBL	Inhibition of ligand binding to Cholecystokinin type A receptor from rat pancreatic tissue.	B	5.8	pIC50	1600	nM	IC50	J. Med. Chem. (1997) 40: 2491-2501 [PMID:9258356]
CCK2 receptor/Cholecystokinin B receptor in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL298] [GtoPdb: 77] [UniProtKB: P32239]
GtoPdb	-	-	9.2	pIC50	0.63	nM	IC50	Regul Pept (2002) 103: 29-37 [PMID:11738246]
ChEMBL	Displacement of [125I]-BH CCK-8S from Cholecystokinin type B receptor in guinea pig cortex	B	10	pIC50	0.1	nM	IC50	Bioorg. Med. Chem. Lett. (1995) 5: 3023-3026
ChEMBL	Inhibition of ligand binding to Cholecystokinin type B receptor from guinea pig cortical membrane.	B	10	pIC50	0.1	nM	IC50	J. Med. Chem. (1997) 40: 2491-2501 [PMID:9258356]

ChEMBL data shown on this page come from version 31:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, Cibrián-Uhalte E, Davies M, Dedman N, Karlsson A, Magariños MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]