ChEMBL ligand: CHEMBL16044
nicotinic acetylcholine receptor δ subunit/Acetylcholine receptor protein delta chain in Human [ChEMBL: CHEMBL3011] [GtoPdb: 476] [UniProtKB: Q07001] There should be some charts here, you may need to enable JavaScript!

DB	Assay description	Assay Type	Standard value	Standard parameter	Original value	Original units	Original parameter	Reference
nicotinic acetylcholine receptor δ subunit/Acetylcholine receptor protein delta chain in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL3011] [GtoPdb: 476] [UniProtKB: Q07001]
ChEMBL	Compound was evaluated for inhibitory activity against human embryonic muscle type Nicotinic acetylcholine receptor specifically delta-subunit expressed in TE-671 cell (at holding potential -50 mV)	B	6.24	pIC50	580	nM	IC50	Bioorg Med Chem Lett (2002) 12: 1159-1162 [PMID:11934578]
ChEMBL	Compound was evaluated for inhibitory activity against human embryonic muscle type Nicotinic acetylcholine receptor specifically delta-subunit expressed in TE-671 cell (at holding potential -100 mV)	B	6.34	pIC50	460	nM	IC50	Bioorg Med Chem Lett (2002) 12: 1159-1162 [PMID:11934578]
GtoPdb	-	-	6.34	pIC50	460	nM	IC50	Bioorg Med Chem Lett (2002) 12: 1159-62 [PMID:11934578]

ChEMBL data shown on this page come from version 34:

Zdrazil B, Felix E, Hunter F, Manners EJ, Blackshaw J, Corbett S, de Veij M, Ioannidis H, Lopez DM, Mosquera JF, Magarinos MP, Bosc N, Arcila R, Kizilören T, Gaulton A, Bento AP, Adasme MF, Monecke P, Landrum GA, Leach AR. (2024). The ChEMBL Database in 2023: a drug discovery platform spanning multiple bioactivity data types and time periods. Nucleic Acids Res., 52(D1). DOI: 10.1093/nar/gkad1004. [EPMCID:10767899] [PMID:37933841]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]