BIA 10-2474 [Ligand Id: 9001] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| Fatty acid amide hydrolase in Human [GtoPdb: 1400] [UniProtKB: O00519] | ||||||||
| GtoPdb | Inhibition of human FAAH expressed in HEK293T cells. | - | 7.3 | pIC50 | 50 | nM | IC50 | Science (2017) 356: 1084-1087 [PMID:28596366] |
| Fatty acid amide hydrolase in Rat [GtoPdb: 1400] [UniProtKB: P97612] | ||||||||
| GtoPdb | This value is an extrapolated estimate from % inhibition data provided in Table 1 of the referenced patent. | - | 6.7 | pIC50 | ~200 | nM | IC50 | WO2010074588 A2. Pharmaceutical compounds. (2010) |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
