ulixertinib [Ligand Id: 9210] activity data from GtoPdb

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  • mitogen-activated protein kinase 3 in Human [GtoPdb: 1494] [UniProtKB: P27361]
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  • mitogen-activated protein kinase 1 in Human [GtoPdb: 1495] [UniProtKB: P28482]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
mitogen-activated protein kinase 3 in Human [GtoPdb: 1494] [UniProtKB: P27361]
GtoPdb Biochemical assay determination - 9.52 pIC50 <0.3 nM IC50 J Med Chem (2015) 58: 4790-801 [PMID:25977981]
mitogen-activated protein kinase 1 in Human [GtoPdb: 1495] [UniProtKB: P28482]
GtoPdb Biochemical assay determination - 9.52 pIC50 <0.3 nM IC50 J Med Chem (2015) 58: 4790-801 [PMID:25977981]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.