compound 6j [PMID: 27219676] [Ligand Id: 9230] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| discoidin domain receptor tyrosine kinase 1 in Human [GtoPdb: 1843] [UniProtKB: Q08345] | ||||||||
| GtoPdb | Binding affinity | - | 8.33 | pKd | 4.7 | nM | Kd | J Med Chem (2016) 59: 5911-6 [PMID:27219676] |
| GtoPdb | Inhibition of kinase activity in a TR-FRET assay | - | 8.03 | pIC50 | 9.4 | nM | IC50 | J Med Chem (2016) 59: 5911-6 [PMID:27219676] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
