AZ3451 [Ligand Id: 9560] activity data from GtoPdb

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  • PAR2 in Human [GtoPdb: 348] [UniProtKB: P55085]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
PAR2 in Human [GtoPdb: 348] [UniProtKB: P55085]
GtoPdb In a BIACORE assay. - 7.87 pKd 13.5 nM Kd Nature (2017) 545: 112-115 [PMID:28445455]
GtoPdb Antagonism of SLIGRL-NH2-induced IP1 formation. - 7.64 pIC50 23 nM IC50 Nature (2017) 545: 112-115 [PMID:28445455]
GtoPdb In a FLIPR calcium accumulation assay, vs. SLIGRL activation. - 8.27 pIC50 5.4 nM IC50 Nature (2017) 545: 112-115 [PMID:28445455]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.