compound 8c [PMID: 28760529] [Ligand Id: 9671] activity data from GtoPdb

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  • BCL6 transcription repressor in Human [GtoPdb: 2957] [UniProtKB: P41182]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
BCL6 transcription repressor in Human [GtoPdb: 2957] [UniProtKB: P41182]
GtoPdb In a cell-based mammalian two-hybrid system assessing inhibition of protein-protein interaction between BCL6 BTB domain and BCoR. - 6.14 pIC50 720 nM IC50 Bioorg Med Chem (2017) 25: 4876-4886 [PMID:28760529]
GtoPdb In a cell-free ELISA system measuring ability to inhibit BCL6 BTB domain-NCoR interaction. - 7 pIC50 100 nM IC50 Bioorg Med Chem (2017) 25: 4876-4886 [PMID:28760529]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.