conteltinib [Ligand Id: 9763] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| protein tyrosine kinase 2 in Human [GtoPdb: 2180] [UniProtKB: Q05397] | ||||||||
| GtoPdb | In a time-resolved fluorescence (TRF) assay using recombinant GST-tagged FAK. | - | 7.7 | pIC50 | <20 | nM | IC50 | WO2012092880. 2,4-DIAMINO-6,7-DIHYDRO-5H-PYRROLO[2,3]PYRIMIDINE DERIVATIVES AS FAK/Pyk2 INHIBITORS (2012) |
| protein tyrosine kinase 2 beta in Human [GtoPdb: 2181] [UniProtKB: Q14289] | ||||||||
| GtoPdb | In a time-resolved fluorescence (TRF) assay using recombinant GST-tagged Pyk2. | - | 7.7 | pIC50 | <20 | nM | IC50 | WO2012092880. 2,4-DIAMINO-6,7-DIHYDRO-5H-PYRROLO[2,3]PYRIMIDINE DERIVATIVES AS FAK/Pyk2 INHIBITORS (2012) |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
