Galapagos MAPKAPK5 inhibitor D [Ligand Id: 9848] activity data from GtoPdb

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  • MAPK activated protein kinase 5 in Human [GtoPdb: 2096] [UniProtKB: Q8IW41]
  • This target only has 0 pki data point
1 _lig_chart_1 MAPK activated protein kinase 5 Human
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
MAPK activated protein kinase 5 in Human [GtoPdb: 2096] [UniProtKB: Q8IW41]
GtoPdb - - 7.43 pIC50 37 nM IC50 Discovery of inhibitors of MAPKAPK5, a novel target for rheumatoid arthritis.
GtoPdb Binned IC50 range from patent. - 9 pIC50 1 nM IC50 WO2007138072A2. Triazolopyrazine compounds useful for the treatment of degenerative & inflammatory diseases (2007)

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.