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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| Bruton tyrosine kinase in Human [GtoPdb: 1948] [UniProtKB: Q06187] | ||||||||
| GtoPdb | Biochemical assay result. Binned IC50 value provided in patent. | - | 7.3 | pIC50 | <50 | nM | IC50 | WO2011162515A2. Novel fused pyrimidine derivatives for inhd3ition of tyrosine kinase activity. (2011) |
| Janus kinase 3 in Human [GtoPdb: 2049] [UniProtKB: P52333] | ||||||||
| GtoPdb | Biochemical assay result. Binned IC50 value provided in patent. | - | 7.3 | pIC50 | <50 | nM | IC50 | WO2011162515A2. Novel fused pyrimidine derivatives for inhd3ition of tyrosine kinase activity. (2011) |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.