xiliertinib [Ligand Id: 9929] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| epidermal growth factor receptor in Human [GtoPdb: 1797] [UniProtKB: P00533] | ||||||||
| GtoPdb | - | - | 10.3 | pKi | 0.05 | nM | Ki | Oncotarget (2017) 8: 50832-50844 [PMID:28881608] |
| erb-b2 receptor tyrosine kinase 4 in Human [GtoPdb: 1799] [UniProtKB: Q15303] | ||||||||
| GtoPdb | - | - | 6.15 | pIC50 | 705 | nM | IC50 | Oncotarget (2017) 8: 50832-50844 [PMID:28881608] |
| LCK proto-oncogene, Src family tyrosine kinase in Human [GtoPdb: 2053] [UniProtKB: P06239] | ||||||||
| GtoPdb | - | - | 6.75 | pIC50 | 176 | nM | IC50 | Oncotarget (2017) 8: 50832-50844 [PMID:28881608] |
| LYN proto-oncogene, Src family tyrosine kinase in Human [GtoPdb: 2060] [UniProtKB: P07948] | ||||||||
| GtoPdb | - | - | 6.3 | pIC50 | 501 | nM | IC50 | Oncotarget (2017) 8: 50832-50844 [PMID:28881608] |
| tyrosine kinase non receptor 1 in Human [GtoPdb: 2245] [UniProtKB: Q13470] | ||||||||
| GtoPdb | - | - | 6.59 | pIC50 | 256 | nM | IC50 | Oncotarget (2017) 8: 50832-50844 [PMID:28881608] |
| YES proto-oncogene 1, Src family tyrosine kinase in Human [GtoPdb: 2284] [UniProtKB: P07947] | ||||||||
| GtoPdb | - | - | 6.48 | pIC50 | 334 | nM | IC50 | Oncotarget (2017) 8: 50832-50844 [PMID:28881608] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
