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edotreotide   Click here for help

GtoPdb Ligand ID: 5638

Synonyms: DOTA-Tyr3-octreotide | DOTA0-Phe1-Tyr3-octreotide | Ga-DOTA-TOC | Ga-DOTATOC | SMT487 | SomaKit TOC®
Approved drug
edotreotide is an approved drug (EMA (2016))
Compound class: Peptide
Comment: Edotreotide is somatostatin receptor agonist. It is radiolabelled with gallium (68Ga) chloride for PET imaging.
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Selectivity at GPCRs
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Target Sp. Type Action Value Parameter Concentration range (M) Reference
SST2 receptor Hs Agonist Full agonist 8.6 pIC50 - 1
pIC50 8.6 (IC50 2.5x10-9 M) [1]