GtoPdb Ligand ID: 6959

Synonyms: (3E)-hex-3-enoylsomatoliberin | Egrifta® | TH9507
tesamorelin is an approved drug (FDA (2010))
Comment: This drug is a stabilized synthetic peptide analogue of the hypothalamic peptide GHRH. The approved formulation is the acetate salt. As with many peptide molecules there is some ambiguity in the literature and on online rescources as to the exact structure and stereochemistry of tesamorelin, therefore we have chosen not to include a chemical structure here. Please see the links above to PubChem, ChEMBL and ChEBI for alternative representations of the structure.
Compound class Peptide or derivative
Approved drug? Yes (FDA (2010))
International Nonproprietary Names
INN number INN
8786 tesamorelin
(3E)-hex-3-enoylsomatoliberin | Egrifta® | TH9507
Database Links
CAS Registry No. 218949-48-5 (source: Scifinder)
ChEMBL Ligand CHEMBL1237026
DrugBank Ligand DB08869
GtoPdb PubChem SID 178103540
PubChem CID 16137828
Search PubMed clinical trials tesamorelin
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Wikipedia Tesamorelin