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bromodomain and PHD finger containing 3

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Target not currently curated in GtoImmuPdb

Target id: 2731

Nomenclature: bromodomain and PHD finger containing 3

Family: Non-enzymatic BRD containing proteins

Gene and Protein Information Click here for help
Species TM AA Chromosomal Location Gene Symbol Gene Name Reference
Human - 1205 6p21.31 BRPF3 bromodomain and PHD finger containing 3
Mouse - 1204 17 A3.3 Brpf3 bromodomain and PHD finger containing, 3
Rat - 1199 20p12 Brpf3 bromodomain and PHD finger containing, 3
Previous and Unofficial Names Click here for help
bromodomain and PHD finger containing, 3 | bromodomain and PHD finger containing
Database Links Click here for help
CATH/Gene3D
ChEMBL Target
Ensembl Gene
Entrez Gene
Human Protein Atlas
KEGG Gene
Pharos
RefSeq Nucleotide
RefSeq Protein
UniProtKB
Wikipedia
Other Binding Ligands
Key to terms and symbols Click column headers to sort
Ligand Sp. Action Value Parameter Reference
NI-57 Small molecule or natural product Click here for species-specific activity table Ligand has a PDB structure Hs Binding 6.4 pKd 2
pKd 6.4 (Kd 4.08x10-7 M) [2]
OF-1 Small molecule or natural product Click here for species-specific activity table Ligand has a PDB structure Hs Binding 5.6 pKd 1
pKd 5.6 (Kd 2.4x10-6 M) [1]
Description: By isothermal titration calorimetry.

References

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1. SGC. OF-1 A chemical probe for BRPF bromodomains. Accessed on 05/04/2017. Modified on 05/04/2017. SGC, http://www.thesgc.org/chemical-probes/OF-1

2. Structural Genomics Consortium. NI-57 – a chemical probe for BRPF bromodomains. Accessed on 15/07/2015. Modified on 15/07/2015. http://www.thesgc.org, http://www.thesgc.org/chemical-probes/NI-57

How to cite this page

Non-enzymatic BRD containing proteins: bromodomain and PHD finger containing 3. Last modified on 05/04/2017. Accessed on 27/11/2020. IUPHAR/BPS Guide to PHARMACOLOGY, http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=2731.