VCE-004.3 [Ligand Id: 10030] activity data from GtoPdb

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  • CB1 receptor in Human [GtoPdb: 56] [UniProtKB: P21554]
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  • CB2 receptor in Human [GtoPdb: 57] [UniProtKB: P34972]
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  • Peroxisome proliferator-activated receptor-γ in Human [GtoPdb: 595] [UniProtKB: P37231]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
CB1 receptor in Human [GtoPdb: 56] [UniProtKB: P21554]
GtoPdb - - 5.61 pKi 2454 nM Ki Br J Pharmacol (2018) 175: 3813-3831 [PMID:30033591]
CB2 receptor in Human [GtoPdb: 57] [UniProtKB: P34972]
GtoPdb - - 6.69 pKi 204 nM Ki Br J Pharmacol (2018) 175: 3813-3831 [PMID:30033591]
Peroxisome proliferator-activated receptor-γ in Human [GtoPdb: 595] [UniProtKB: P37231]
GtoPdb - - 5.46 pIC50 3500 nM IC50 Br J Pharmacol (2018) 175: 3813-3831 [PMID:30033591]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.