azelaprag [Ligand Id: 10061] activity data from GtoPdb

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  • apelin receptor in Human [GtoPdb: 36] [UniProtKB: P35414]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
apelin receptor in Human [GtoPdb: 36] [UniProtKB: P35414]
GtoPdb Measuring ligand-induced [35S]GTPyS Binding in membranes prepared fron CHO cells stably expressing human apelin receptor. - 9.49 pEC50 0.32 nM EC50 WO2016187308A1. Triazole agonists of the apj receptor (2016)

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.