PFKFB3 kinase Inhibitor 69 [Ligand Id: 10125] activity data from GtoPdb
Click here for a description of the charts and data table
Please tell us if you are using this feature and what you think!
|
There should be some charts here, you may need to enable JavaScript!
|
| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| 6-phosphofructo-2-kinase/fructose-2,6-biphosphatase 3 in Human [GtoPdb: 2937] [UniProtKB: Q16875] | ||||||||
| GtoPdb | In a biochemical assay using purified recombinant human His-tagged PFKFB3, and the production of ADP as readout (ADP-Glo™ Kinase Assay kit from Promega) | - | 7.85 | pIC50 | 14 | nM | IC50 | ChemMedChem (2019) 14: 169-181 [PMID:30378281] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
