AM10257 [Ligand Id: 10177] activity data from GtoPdb

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  • CB2 receptor in Human [GtoPdb: 57] [UniProtKB: P34972]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
CB2 receptor in Human [GtoPdb: 57] [UniProtKB: P34972]
GtoPdb Antagonism of [3H]CP55940 binding to human CB2. - 10.12 pKi 0.08 nM Ki Cell (2019) 176: 459-467.e13 [PMID:30639103]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.