linperlisib [Ligand Id: 10466] activity data from GtoPdb

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  • phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit delta in Human [GtoPdb: 2155] [UniProtKB: O00329]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit delta in Human [GtoPdb: 2155] [UniProtKB: O00329]
GtoPdb Measured in a luminescence assay to detect modulation of ADP formation in the presence of test compound and hPI3Kδ. - 8.62 pIC50 2.4 nM IC50 US20160244432A1. Fused heterocyclic compound, preparation method therefor, pharmaceutcial composition, and uses thereof (2017)

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.