bamocaftor [Ligand Id: 10553] activity data from GtoPdb

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  • CFTR in Human [GtoPdb: 707] [UniProtKB: P13569]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
CFTR in Human [GtoPdb: 707] [UniProtKB: P13569]
GtoPdb - - 7.52 pEC50 30 nM EC50 N Engl J Med (2018) 379: 1599-1611 [PMID:30334693];
WO2018064632A1. Modulator of cystic fibrosis transmembrane conductance regulator, pharmaceutical compositions, methods of treatment, and process for making the modulator (2018)

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.