compound 32 [PMID: 31675166] [Ligand Id: 10576] activity data from GtoPdb

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  • kallikrein related peptidase 4 in Human [GtoPdb: 2374] [UniProtKB: Q9Y5K2]
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  • kallikrein related peptidase 6 in Human [GtoPdb: 2376] [UniProtKB: Q92876]
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  • kallikrein related peptidase 8 in Human [GtoPdb: 2378] [UniProtKB: O60259]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
kallikrein related peptidase 4 in Human [GtoPdb: 2374] [UniProtKB: Q9Y5K2]
GtoPdb - - 6.8 pIC50 158 nM IC50 ChemMedChem (2020) 15: 79-95 [PMID:31675166]
kallikrein related peptidase 6 in Human [GtoPdb: 2376] [UniProtKB: Q92876]
GtoPdb - - 8.6 pIC50 2.5 nM IC50 ChemMedChem (2020) 15: 79-95 [PMID:31675166]
kallikrein related peptidase 8 in Human [GtoPdb: 2378] [UniProtKB: O60259]
GtoPdb - - 6.7 pIC50 200 nM IC50 ChemMedChem (2020) 15: 79-95 [PMID:31675166]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.