JNJ-42226314 [Ligand Id: 10661] activity data from GtoPdb

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  • Monoacylglycerol lipase in Human [GtoPdb: 1399] [UniProtKB: Q99685]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
Monoacylglycerol lipase in Human [GtoPdb: 1399] [UniProtKB: Q99685]
GtoPdb In vitro potency of JNJ-42226314 to inhibit human MAGL using an in vitro [3H]2-OG cleavage activity assay. - 8.95 pIC50 1.13 nM IC50 J. Pharmacol. Exp. Ther. (2020) 372: 339-353 [PMID:31818916]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.