(R)-16 [PMID: 32267688] [Ligand Id: 10751] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| Peroxisome proliferator-activated receptor-α in Human [GtoPdb: 593] [UniProtKB: Q07869] | ||||||||
| GtoPdb | Measuring nuclear receptor modulation in Gal4-hybrid reporter gene assays conducted in transiently transfected HEK293T cells. | - | 6.37 | pEC50 | 430 | nM | EC50 | J Med Chem (2020) 63: 4555-4561 [PMID:32267688] |
| Peroxisome proliferator-activated receptor-β/δ in Human [GtoPdb: 594] [UniProtKB: Q03181] | ||||||||
| GtoPdb | Measuring nuclear receptor modulation in Gal4-hybrid reporter gene assays conducted in transiently transfected HEK293T cells. | - | 6.09 | pEC50 | 810 | nM | EC50 | J Med Chem (2020) 63: 4555-4561 [PMID:32267688] |
| Peroxisome proliferator-activated receptor-γ in Human [GtoPdb: 595] [UniProtKB: P37231] | ||||||||
| GtoPdb | Measuring nuclear receptor modulation in Gal4-hybrid reporter gene assays conducted in transiently transfected HEK293T cells. | - | 8.8 | pEC50 | 1.6 | nM | EC50 | J Med Chem (2020) 63: 4555-4561 [PMID:32267688] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
