DCLK1-IN-1 [Ligand Id: 11114] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| doublecortin like kinase 1 in Human [GtoPdb: 2005] [UniProtKB: O15075] | ||||||||
| GtoPdb | Determined in an ITC assay. | - | 6.96 | pKd | 109 | nM | Kd | Nat Chem Biol (2020) 16: 635-643 [PMID:32251410] |
| GtoPdb | Determined in a NanoBRET cell assay. | - | 6.55 | pIC50 | 279 | nM | IC50 | Nat Chem Biol (2020) 16: 635-643 [PMID:32251410] |
| GtoPdb | Determined in a KinomeScan binding assay. | - | 8.02 | pIC50 | 9.5 | nM | IC50 | Nat Chem Biol (2020) 16: 635-643 [PMID:32251410] |
| doublecortin like kinase 2 in Human [GtoPdb: 2006] [UniProtKB: Q8N568] | ||||||||
| GtoPdb | Determined in a KinomeScan binding assay. | - | 7.51 | pIC50 | 31 | nM | IC50 | Nat Chem Biol (2020) 16: 635-643 [PMID:32251410] |
| leucine rich repeat kinase 2 in Human [GtoPdb: 2059] [UniProtKB: Q5S007] | ||||||||
| GtoPdb | Determined in a LRRK2 ADAPTA kinase assay. | - | 5.16 | pIC50 | 6970 | nM | IC50 | Nat Chem Biol (2020) 16: 635-643 [PMID:32251410] |
| mitogen-activated protein kinase 7 in Human [GtoPdb: 2093] [UniProtKB: Q13164] | ||||||||
| GtoPdb | Determined in a KinomeScan binding assay. | - | 5.74 | pIC50 | 1800 | nM | IC50 | Nat Chem Biol (2020) 16: 635-643 [PMID:32251410] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
