bindarit [Ligand Id: 11124] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL2107549 (Bindarit, AF-2838)
  • fatty acid binding protein 4 in Human [GtoPdb: 2534] [UniProtKB: P15090]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
fatty acid binding protein 4 in Human [GtoPdb: 2534] [UniProtKB: P15090]
GtoPdb Measuring displacement of [3H]-oleic acid from hFABP4 in a competitive binding assay. - 4.72 pKi 19000 nM Ki Sci Rep (2019) 9: 15155 [PMID:31641194]

ChEMBL data shown on this page come from version 27:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, CibriƔn-Uhalte E, Davies M, Dedman N, Karlsson A, MagariƱos MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]