imaradenant [Ligand Id: 11153] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| A1 receptor in Human [GtoPdb: 18] [UniProtKB: P30542] | ||||||||
| GtoPdb | Binding affinity of AZD4635 determined in a radioligand binding competition assays with membranes prepared from CHO cells stably expressing human A1R. | - | 6.8 | pKi | 160 | nM | Ki | J Immunother Cancer (2020) 8: e000417 [PMID:32727810] |
| A2A receptor in Human [GtoPdb: 19] [UniProtKB: P29274] | ||||||||
| GtoPdb | Binding affinity of AZD4635 determined in a radioligand binding competition assays with membranes prepared from HEK-293-T cells stably expressing human A2AR. | - | 8.77 | pKi | 1.7 | nM | Ki | J Immunother Cancer (2020) 8: e000417 [PMID:32727810] |
| A2B receptor in Human [GtoPdb: 20] [UniProtKB: P29275] | ||||||||
| GtoPdb | Binding affinity of AZD4635 determined in a radioligand binding competition assays with membranes prepared from HEK-293-T cells stably expressing human A2BR. | - | 7.19 | pKi | 64 | nM | Ki | J Immunother Cancer (2020) 8: e000417 [PMID:32727810] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
