ChEMBL ligand: CHEMBL1929396 (Anagliptin, CWP-403, Sk-0403, SK-0403, Suiny)
fibroblast activation protein alpha/Fibroblast activation protein alpha in Human [ChEMBL: CHEMBL4683] [GtoPdb: 2365] [UniProtKB: Q12884] There should be some charts here, you may need to enable JavaScript!
dipeptidyl peptidase 4 in Human [GtoPdb: 1612] [UniProtKB: P27487] There should be some charts here, you may need to enable JavaScript!

DB	Assay description	Assay Type	Standard value	Standard parameter	Original value	Original units	Original parameter	Reference
fibroblast activation protein alpha/Fibroblast activation protein alpha in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL4683] [GtoPdb: 2365] [UniProtKB: Q12884]
ChEMBL	Inhibition of human recombinant FAP expressed in baculovirus-infected Sf9 insect cells using H-Ala-Pro-AFC as substrate after 60 mins by fluorescence assay	B	4.14	pIC50	72700	nM	IC50	Bioorg. Med. Chem. (2011) 19: 7221-7227 [PMID:22019046]
dipeptidyl peptidase 4 in Human [GtoPdb: 1612] [UniProtKB: P27487]
GtoPdb	Inhibition of human recombinant DPP-4 in vitro	-	8.42	pIC50	3.8	nM	IC50	Bioorg Med Chem (2011) 19: 7221-7 [PMID:22019046]

ChEMBL data shown on this page come from version 31:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, Cibrián-Uhalte E, Davies M, Dedman N, Karlsson A, Magariños MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]