tinengotinib [Ligand Id: 11887] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| fibroblast growth factor receptor 1 in Human [GtoPdb: 1808] [UniProtKB: P11362] | ||||||||
| GtoPdb | - | - | 8.64 | pIC50 | 2.3 | nM | IC50 | US10889586B2. Multi-kinase inhibitor compound, and crystal form and use thereof (2021) |
| fibroblast growth factor receptor 3 in Human [GtoPdb: 1810] [UniProtKB: P22607] | ||||||||
| GtoPdb | - | - | 8.46 | pIC50 | 3.5 | nM | IC50 | US10889586B2. Multi-kinase inhibitor compound, and crystal form and use thereof (2021) |
| fms related receptor tyrosine kinase 1 in Human [GtoPdb: 1812] [UniProtKB: P17948] | ||||||||
| GtoPdb | - | - | 8.62 | pIC50 | 2.4 | nM | IC50 | US10889586B2. Multi-kinase inhibitor compound, and crystal form and use thereof (2021) |
| kinase insert domain receptor in Human [GtoPdb: 1813] [UniProtKB: P35968] | ||||||||
| GtoPdb | - | - | 8.6 | pIC50 | 2.5 | nM | IC50 | US10889586B2. Multi-kinase inhibitor compound, and crystal form and use thereof (2021) |
| aurora kinase A in Human [GtoPdb: 1936] [UniProtKB: O14965] | ||||||||
| GtoPdb | - | - | 8.92 | pIC50 | 1.2 | nM | IC50 | US10889586B2. Multi-kinase inhibitor compound, and crystal form and use thereof (2021) |
| aurora kinase B in Human [GtoPdb: 1937] [UniProtKB: Q96GD4] | ||||||||
| GtoPdb | - | - | 8.48 | pIC50 | 3.3 | nM | IC50 | US10889586B2. Multi-kinase inhibitor compound, and crystal form and use thereof (2021) |
| Janus kinase 2 in Human [GtoPdb: 2048] [UniProtKB: O60674] | ||||||||
| GtoPdb | - | - | 9.12 | pIC50 | 0.75 | nM | IC50 | US10889586B2. Multi-kinase inhibitor compound, and crystal form and use thereof (2021) |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
