compound 17 [PMID: 36111834] [Ligand Id: 12185] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| myosin light chain kinase family member 4 in Human [GtoPdb: 2111] [UniProtKB: Q86YV6] | ||||||||
| GtoPdb | Determined in a cell-based NanoBRET assay | - | 6.58 | pIC50 | 265 | nM | IC50 | J Med Chem (2022) 65: 12860-12882 [PMID:36111834] |
| phosphoinositide kinase, FYVE-type zinc finger containing in Human [GtoPdb: 2857] [UniProtKB: Q9Y2I7] | ||||||||
| GtoPdb | Inhibition of hPIKFYVE in a proprietary ADP-Glo enzymatic assay | - | 8.16 | pIC50 | 6.9 | nM | IC50 | J Med Chem (2022) 65: 12860-12882 [PMID:36111834] |
| GtoPdb | Determined in a cell-based NanoBRET assay | - | 8.4 | pIC50 | 4.01 | nM | IC50 | J Med Chem (2022) 65: 12860-12882 [PMID:36111834] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
