zongertinib [Ligand Id: 12387] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| epidermal growth factor receptor in Human [GtoPdb: 1797] [UniProtKB: P00533] | ||||||||
| GtoPdb | Inhibition of wild type EGFR phosphorylation | - | 6.24 | pIC50 | 579 | nM | IC50 | WO2021156178A1. [1,3]diazino[5,4-d]pyrimidines as her2 inhibitors (2021) |
| erb-b2 receptor tyrosine kinase 2 in Human [GtoPdb: 2019] [UniProtKB: P04626] | ||||||||
| GtoPdb | Inhibition of phosphorylation of HER2 YMVA mutation | - | 7.89 | pIC50 | 13 | nM | IC50 | WO2021156178A1. [1,3]diazino[5,4-d]pyrimidines as her2 inhibitors (2021) |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
