I-BET282 [Ligand Id: 12717] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| bromodomain containing 4 in Human [GtoPdb: 1945] [UniProtKB: O60885] | ||||||||
| GtoPdb | Inhibition of BRD4 BD1 | - | 7.4 | pIC50 | 39.4 | nM | IC50 | J Med Chem (2021) 64: 12200-12227 [PMID:34387088] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
