ChEMBL ligand: CHEMBL3330226 (Macozinona, Macozinone, PBTZ-169, PBTZ169)
FAD-dependent decaprenylphosphoryl-beta-D-ribofuranose 2-oxidase in Mycobacterium tuberculosis [ChEMBL: CHEMBL3804751] [UniProtKB: P9WJF1] There should be some charts here, you may need to enable JavaScript!

DB	Assay description	Assay Type	Standard value	Standard parameter	Original value	Original units	Original parameter	Reference
FAD-dependent decaprenylphosphoryl-beta-D-ribofuranose 2-oxidase in Mycobacterium tuberculosis (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL3804751] [UniProtKB: P9WJF1]
ChEMBL	Inhibition of Mycobacterium tuberculosis DprE1 expressed in Escherichia coli BL21 (DE3) cells assessed as formation of resorufin using FPR as substrate by Amplex Red hydrogen/peroxidase coupled assay	B	8	pIC50	10	nM	IC50	Eur J Med Chem (2020) 208: 112773-112773 [PMID:32898793]
ChEMBL	Inhibition of Mycobacterium tuberculosis H37Rv recombinant DprE1 expressed in Escherichia coli assessed as formation of resorufin using FPR as substrate by Amplex Red hydrogen/peroxidase coupled assay	B	8	pIC50	10	nM	IC50	ACS Med Chem Lett (2022) 13: 593-598 [PMID:35450361]

ChEMBL data shown on this page come from version 34:

Zdrazil B, Felix E, Hunter F, Manners EJ, Blackshaw J, Corbett S, de Veij M, Ioannidis H, Lopez DM, Mosquera JF, Magarinos MP, Bosc N, Arcila R, Kizilören T, Gaulton A, Bento AP, Adasme MF, Monecke P, Landrum GA, Leach AR. (2024). The ChEMBL Database in 2023: a drug discovery platform spanning multiple bioactivity data types and time periods. Nucleic Acids Res., 52(D1). DOI: 10.1093/nar/gkad1004. [EPMCID:10767899] [PMID:37933841]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]