monlunabant [Ligand Id: 13717] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| CB1 receptor in Human [GtoPdb: 56] [UniProtKB: P21554] | ||||||||
| GtoPdb | Measuring inhibition of [3H]CP55940 (agonist) binding to CB1 receptor | - | 9.52 | pKi | 0.3 | nM | Ki | ACS Pharmacol Transl Sci (2021) 4: 1175-1187 [PMID:34151207] |
| GtoPdb | Determined in a GTPγS assay | - | 8.22 | pIC50 | 6 | nM | IC50 | ACS Pharmacol Transl Sci (2021) 4: 1175-1187 [PMID:34151207] |
| GtoPdb | Determined in a βArr2 recruitment assay | - | 10.68 | pIC50 | 0.02 | nM | IC50 | ACS Pharmacol Transl Sci (2021) 4: 1175-1187 [PMID:34151207] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
