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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference | 
|---|---|---|---|---|---|---|---|---|
| ret proto-oncogene in Human [GtoPdb: 2185] [UniProtKB: P07949] | ||||||||
| GtoPdb | Potency for RET V804M | - | 9.9 | pIC50 | 0.13 | nM | IC50 | J Med Chem (2025) : [PMID:40920215] | 
| GtoPdb | Potenct for WT RET | - | 10.02 | pIC50 | 0.09 | nM | IC50 | J Med Chem (2025) : [PMID:40920215] | 
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.