nomelcitinib [Ligand Id: 14360] activity data from GtoPdb

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  • tyrosine kinase 2 in Human [GtoPdb: 2269] [UniProtKB: P29597]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
tyrosine kinase 2 in Human [GtoPdb: 2269] [UniProtKB: P29597]
GtoPdb Measuring inhibition of IL-23-mediate STAT3 pathway activation in HEK-Blue IL23 cells - 8.6 pIC50 2.5 nM IC50 WO2022135430A1. Heteroaryl compounds, preparation methods and uses thereof (2022)

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.