C4Pen [Ligand Id: 14460] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| Nav1.2 in Human [GtoPdb: 579] [UniProtKB: Q99250] | ||||||||
| GtoPdb | - | - | 7.48 | pIC50 | 33.12 | nM | IC50 | J Med Chem (2026) : |
| Nav1.4 in Human [GtoPdb: 581] [UniProtKB: P35499] | ||||||||
| GtoPdb | - | - | 7.95 | pIC50 | 11.1 | nM | IC50 | J Med Chem (2026) : |
| Nav1.7 in Human [GtoPdb: 584] [UniProtKB: Q15858] | ||||||||
| GtoPdb | - | - | 7.11 | pIC50 | 77.4 | nM | IC50 | J Med Chem (2026) : |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
