bilobalide [Ligand Id: 2366] activity data from GtoPdb and ChEMBL
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| ChEMBL ligand: CHEMBL1318117 |
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| 5-HT3AB in Human [GtoPdb: 378] | ||||||||
| GtoPdb | - | - | 2.51 | pIC50 | 3100000 | nM | IC50 | Neuropharmacology (2011) 60: 488-95 [PMID:21059362] |
| 5-HT3A in Human [GtoPdb: 379] | ||||||||
| GtoPdb | - | - | 3.33 | pIC50 | 470000 | nM | IC50 | Mol Pharmacol (2011) 80: 183-90 [PMID:21505038] |
| glycine receptor α1 subunit in Human [GtoPdb: 423] [UniProtKB: P23415] | ||||||||
| GtoPdb | - | - | 4.7 | pIC50 | 20000 | nM | IC50 | |
| glycine receptor α2 subunit in Human [GtoPdb: 424] [UniProtKB: P23416] | ||||||||
| GtoPdb | - | - | 5.1 | pIC50 | 8000 | nM | IC50 | |
| glycine receptor β subunit in Human [GtoPdb: 427] [UniProtKB: P48167] | ||||||||
| GtoPdb | - | - | 3.7 | pIC50 | 204000 | nM | IC50 | |
| GtoPdb | - | - | 4.3 | pIC50 | 50000 | nM | IC50 | |
ChEMBL data shown on this page come from version 31:
Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, Cibrián-Uhalte E, Davies M, Dedman N, Karlsson A, Magariños MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]
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