Gd3+ [Ligand Id: 2426] activity data from GtoPdb

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  • TRPA1 in Mouse [GtoPdb: 485] [UniProtKB: Q8BLA8]
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  • TRPC3 in Human [GtoPdb: 488] [UniProtKB: Q13507]
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  • TRPC6 in Mouse [GtoPdb: 491] [UniProtKB: Q61143]
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  • TRPM3 in Human [GtoPdb: 495] [UniProtKB: Q9HCF6]
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  • TRPML3 in Mouse [GtoPdb: 503] [UniProtKB: Q8R4F0]
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  • ASIC3 in Human [GtoPdb: 686] [UniProtKB: Q9UHC3]
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  • Navi2.1 in Human [GtoPdb: 750] [UniProtKB: Q8IZF0]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
TRPA1 in Mouse [GtoPdb: 485] [UniProtKB: Q8BLA8]
GtoPdb - - 7 pIC50 - - - J. Neurosci. (2005) 25: 4052-61 [PMID:15843607]
TRPC3 in Human [GtoPdb: 488] [UniProtKB: Q13507]
GtoPdb - - 7 pEC50 100 nM EC50 J. Biol. Chem. (2000) 275: 37423-8 [PMID:10970899]
TRPC6 in Mouse [GtoPdb: 491] [UniProtKB: Q61143]
GtoPdb - - 5.7 pIC50 1900 nM IC50 Circ. Res. (2001) 88: 325-32 [PMID:11179201]
TRPM3 in Human [GtoPdb: 495] [UniProtKB: Q9HCF6]
GtoPdb - - 4 pIC50 - - - J. Biol. Chem. (2003) 278: 20890-7 [PMID:12672827];
J. Biol. Chem. (2003) 278: 21493-501 [PMID:12672799]
TRPML3 in Mouse [GtoPdb: 503] [UniProtKB: Q8R4F0]
GtoPdb - - 4.7 pIC50 20000 nM IC50 Proc. Natl. Acad. Sci. U.S.A. (2008) 105: 353-8 [PMID:18162548]
ASIC3 in Human [GtoPdb: 686] [UniProtKB: Q9UHC3]
GtoPdb - - 4.4 pIC50 40000 nM IC50
Navi2.1 in Human [GtoPdb: 750] [UniProtKB: Q8IZF0]
GtoPdb - - 5.6 pIC50 1400 nM IC50

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.