Gd3+ [Ligand Id: 2426] activity data from GtoPdb

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  • TRPA1 in Mouse [GtoPdb: 485] [UniProtKB: Q8BLA8]
  • This target only has 0 pki data point
  • 0
1 _lig_chart_1 TRPA1 Mouse
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  • TRPC3 in Human [GtoPdb: 488] [UniProtKB: Q13507]
  • This target only has 0 pki data point
  • 0
2 _lig_chart_2 TRPC3 Human
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  • TRPC6 in Mouse [GtoPdb: 491] [UniProtKB: Q61143]
  • This target only has 0 pki data point
  • 0
3 _lig_chart_3 TRPC6 Mouse
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  • TRPM3 in Human [GtoPdb: 495] [UniProtKB: Q9HCF6]
  • This target only has 0 pki data point
  • 0
4 _lig_chart_4 TRPM3 Human
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  • TRPML3 in Mouse [GtoPdb: 503] [UniProtKB: Q8R4F0]
  • This target only has 0 pki data point
  • 0
5 _lig_chart_5 TRPML3 Mouse
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  • ASIC3 in Human [GtoPdb: 686] [UniProtKB: Q9UHC3]
  • This target only has 0 pki data point
  • 0
6 _lig_chart_6 ASIC3 Human
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  • Navi2.1 in Human [GtoPdb: 750] [UniProtKB: Q8IZF0]
  • This target only has 0 pki data point
  • 0
7 _lig_chart_7 Navi2.1 Human
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
TRPA1 in Mouse [GtoPdb: 485] [UniProtKB: Q8BLA8]
GtoPdb - - 7 pIC50 - - - J Neurosci (2005) 25: 4052-61 [PMID:15843607]
TRPC3 in Human [GtoPdb: 488] [UniProtKB: Q13507]
GtoPdb - - 7 pEC50 100 nM EC50 J Biol Chem (2000) 275: 37423-8 [PMID:10970899]
TRPC6 in Mouse [GtoPdb: 491] [UniProtKB: Q61143]
GtoPdb - - 5.7 pIC50 1900 nM IC50 Circ Res (2001) 88: 325-32 [PMID:11179201]
TRPM3 in Human [GtoPdb: 495] [UniProtKB: Q9HCF6]
GtoPdb - - 4 pIC50 - - - J Biol Chem (2003) 278: 20890-7 [PMID:12672827];
J Biol Chem (2003) 278: 21493-501 [PMID:12672799]
TRPML3 in Mouse [GtoPdb: 503] [UniProtKB: Q8R4F0]
GtoPdb - - 4.7 pIC50 20000 nM IC50 Proc Natl Acad Sci USA (2008) 105: 353-8 [PMID:18162548]
ASIC3 in Human [GtoPdb: 686] [UniProtKB: Q9UHC3]
GtoPdb - - 4.4 pIC50 40000 nM IC50 J Biol Chem (2000) 275: 28519-25 [PMID:10842183]
Navi2.1 in Human [GtoPdb: 750] [UniProtKB: Q8IZF0]
GtoPdb - - 5.6 pIC50 1400 nM IC50

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.