OMPT [Ligand Id: 2912] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL1395060
  • LPA3 receptor/Lysophosphatidic acid receptor Edg-7 in Human [ChEMBL: CHEMBL3250] [GtoPdb: 274] [UniProtKB: Q9UBY5]
  • This target only has 0 pki data point
1 CHEMBL1395060_lig_chart_1 Lysophosphatidic acid receptor Edg-7 Human
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
LPA3 receptor/Lysophosphatidic acid receptor Edg-7 in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL3250] [GtoPdb: 274] [UniProtKB: Q9UBY5]
ChEMBL Agonist activity at human LPA3 receptor transfected in HEK293T cells after 30 mins by GTP[gamma-35S] binding assay B 6.56 pEC50 276 nM EC50 MedChemComm (2015) 6: 13-23
GtoPdb - - 7.17 pEC50 - - - J. Biol. Chem. (2003) 278: 11962-9 [PMID:12554733]

ChEMBL data shown on this page come from version 27:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, CibriƔn-Uhalte E, Davies M, Dedman N, Karlsson A, MagariƱos MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]