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ChEMBL ligand: CHEMBL870 |
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DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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farnesyl diphosphate synthase in Human [GtoPdb: 644] [UniProtKB: P14324] | ||||||||
GtoPdb | - | - | 6.34 | pIC50 | 460 | nM | IC50 | Arch Biochem Biophys (2000) 373: 231-41 [PMID:10620343] |
GtoPdb | In vitro inhibition of recombinant human protein expressed in E coli. | - | 7.3 | pIC50 | 50 | nM | IC50 | J Pharmacol Exp Ther (2001) 296: 235-42 [PMID:11160603] |
ChEMBL data shown on this page come from version 28:
Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, CibriƔn-Uhalte E, Davies M, Dedman N, Karlsson A, MagariƱos MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]