SNAP5089 [Ligand Id: 498] activity data from GtoPdb

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  • α1A-adrenoceptor in Human [GtoPdb: 22] [UniProtKB: P35348]
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  • α1D-adrenoceptor in Human [GtoPdb: 24] [UniProtKB: P25100]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
α1A-adrenoceptor in Human [GtoPdb: 22] [UniProtKB: P35348]
GtoPdb - - 9.4 pKi - - - Pharm Acta Helv (2000) 74: 163-71 [PMID:10812954];
J Med Chem (1995) 38: 1579-81 [PMID:7752182];
J Pharmacol Exp Ther (1997) 281: 1272-83 [PMID:9190863];
Pharmacol Res Perspect (2020) 8: e00602 [PMID:32608144]
α1D-adrenoceptor in Human [GtoPdb: 24] [UniProtKB: P25100]
GtoPdb - - 5.7 pKi - - - Pharmacol Res Perspect (2020) 8: e00602 [PMID:32608144]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.