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ChEMBL ligand: CHEMBL321585 (Docosatetra-7Z,10Z,13Z,16Z-Enoyl Ethanolamide) |
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DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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CB1 receptor/Cannabinoid CB1 receptor in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL218] [GtoPdb: 56] [UniProtKB: P21554] | ||||||||
ChEMBL | Compound was evaluated for its binding affinity towards Cannabinoid receptor 1 [Inactive form(R) of CB1 receptor] | B | 7.46 | pKi | 34.4 | nM | Ki | J. Med. Chem. (2002) 45: 3649-3659 [PMID:12166938] |
CB1 receptor/Cannabinoid CB1 receptor in Rat (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL3571] [GtoPdb: 56] [UniProtKB: P20272] | ||||||||
ChEMBL | In vitro binding affinity was determined against rat brain Cannabinoid receptor 1 | B | 7.46 | pKi | 34.4 | nM | Ki | J. Med. Chem. (1997) 40: 659-667 [PMID:9057852] |
ChEMBL | Binding affinity for cannabinoid receptor 1 | B | 7.47 | pKi | 34 | nM | Ki | J. Med. Chem. (2005) 48: 5059-5087 [PMID:16078824] |
ChEMBL data shown on this page come from version 28:
Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, CibriƔn-Uhalte E, Davies M, Dedman N, Karlsson A, MagariƱos MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]