Ap3a [Ligand Id: 5454] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL407938
  • P2Y1 receptor/Purinergic receptor P2Y1 in Rat [ChEMBL: CHEMBL2497] [GtoPdb: 323] [UniProtKB: P49651]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
P2Y1 receptor/Purinergic receptor P2Y1 in Rat (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL2497] [GtoPdb: 323] [UniProtKB: P49651]
GtoPdb - - 7.22 pEC50 60 nM EC50 J Med Chem (2006) 49: 1980-90 [PMID:16539385]
ChEMBL Activity against rat P2Y1-GFP transfected in HEK293 cells by intracellular calcium increase F 7.22 pEC50 60 nM EC50 J. Med. Chem. (2006) 49: 1980-1990 [PMID:16539385]

ChEMBL data shown on this page come from version 28:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, CibriƔn-Uhalte E, Davies M, Dedman N, Karlsson A, MagariƱos MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]