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ChEMBL ligand: CHEMBL499876 |
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1
CHEMBL499876_lig_chart_1
GPR18
Human
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2
CHEMBL499876_lig_chart_2
GPR55
Human
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DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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GPR18 in Human [GtoPdb: 89] [UniProtKB: Q14330] | ||||||||
GtoPdb | - | - | 6.08 | pEC50 | 835.7 | nM | EC50 | Br J Pharmacol (2012) 165: 2414-24 [PMID:21595653] |
GPR55 in Human [GtoPdb: 109] [UniProtKB: Q9Y2T6] | ||||||||
GtoPdb | - | - | 5.71 | pEC50 | 1944 | nM | EC50 | Br J Pharmacol (2007) 152: 1092-101 [PMID:17876302] |
GtoPdb | - | - | 8.6 | pEC50 | 2.5 | nM | EC50 | Br J Pharmacol (2007) 152: 825-31 [PMID:17704827] |
ChEMBL data shown on this page come from version 28:
Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, CibriƔn-Uhalte E, Davies M, Dedman N, Karlsson A, MagariƱos MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]