PD123319 [Ligand Id: 597] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL321820
  • AT2 receptor in Human [GtoPdb: 35] [UniProtKB: P50052]
  • This target only has 0 pki data point
1 CHEMBL321820_lig_chart_1 AT2 receptor Human
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
AT2 receptor in Human [GtoPdb: 35] [UniProtKB: P50052]
GtoPdb - - 9.2 pKd 0.63 nM Kd Heterogeneity of angiotensin receptor subtypes.. Medicinal Chemistry of the Renin-Angiotensin System. (1994);
Mol. Pharmacol. (1990) 38: 370-7 [PMID:2402226];
J. Cardiovasc. Pharmacol. (1991) 17: 177-84 [PMID:1709220]

ChEMBL data shown on this page come from version 27:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, Cibrián-Uhalte E, Davies M, Dedman N, Karlsson A, Magariños MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]