fexagratinib [Ligand Id: 7707] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| Insulin-like growth factor I receptor in Human [GtoPdb: 1801] [UniProtKB: P08069] | ||||||||
| GtoPdb | - | - | 6.24 | pIC50 | 581 | nM | IC50 | AZD4547.. astrazeneca.com |
| fibroblast growth factor receptor 1 in Human [GtoPdb: 1808] [UniProtKB: P11362] | ||||||||
| GtoPdb | - | - | 9.15 | pIC50 | <0.7 | nM | IC50 |
AZD4547.. astrazeneca.com; Org Biomol Chem (2015) 13: 7643-54 [PMID:26080733] |
| fibroblast growth factor receptor 2 in Human [GtoPdb: 1809] [UniProtKB: P21802] | ||||||||
| GtoPdb | - | - | 8.3 | pIC50 | <5 | nM | IC50 | AZD4547.. astrazeneca.com |
| fibroblast growth factor receptor 3 in Human [GtoPdb: 1810] [UniProtKB: P22607] | ||||||||
| GtoPdb | - | - | 8.3 | pIC50 | <5 | nM | IC50 | AZD4547.. astrazeneca.com |
| fibroblast growth factor receptor 4 in Human [GtoPdb: 1811] [UniProtKB: P22455] | ||||||||
| GtoPdb | - | - | 6.78 | pIC50 | 165 | nM | IC50 | AZD4547.. astrazeneca.com |
| kinase insert domain receptor in Human [GtoPdb: 1813] [UniProtKB: P35968] | ||||||||
| GtoPdb | - | - | 7.62 | pIC50 | 24 | nM | IC50 | AZD4547.. astrazeneca.com |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
